SCHEMBL20182274

SCHEMBL20182274

COc1ncccc1-c1cn(C(C)/C(=C/Nc2ccccc2F)N=N)c2ncnc(N)c12

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EIF2AK3 Q9NZJ5 5/20 0.40
KDR P35968 8/20 0.38
RET P07949 3/20 0.38
TEK Q02763 5/20 0.36
SRC P12931 4/20 0.36
LCK P06239 3/20 0.36
EGFR P00533 1/20 0.36
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
PRKDC P78527 1/20 0.35
SOS1 Q07889 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182288 0.85 EIF2AK3 (0.39) EIF2AK3KDRRETTEKSRC
SCHEMBL20173329 0.82 EIF2AK3 (0.38) EIF2AK3TEKSRCLCK
SCHEMBL20182362 0.81 CFTR (0.40) KDRRETTEKSRCLCK
SCHEMBL20182227 0.81 EGFR (0.36) EIF2AK3KDRRETTEKSRC
SCHEMBL20181916 0.80 CFTR (0.39) EIF2AK3KDRTEKSRCLCK
SCHEMBL20182194 0.80 EIF2AK3 (0.36) EIF2AK3KDRRETTEKSRC
SCHEMBL20182228 0.79 KDR (0.45) KDRTEKSRCLCKEGFR
SCHEMBL20181906 0.79 EIF2AK3 (0.34) EIF2AK3KDRRETTEKSRC
SCHEMBL20182283 0.79 NTRK1 (0.36) KDRRETTEKSRCLCK
SCHEMBL20182241 0.79 KDR (0.46) EIF2AK3KDRTEKSRCLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed