SCHEMBL20182252

SCHEMBL20182252

Nc1ncnc2c1c(-c1ccc(Cl)cc1)c(Br)n2SF

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.43
SRC P12931 4/20 0.43
LCK P06239 4/20 0.43
TEK Q02763 4/20 0.43
FYN P06241 3/20 0.43
CYP1A2 P05177 3/20 0.43
ABL1 P00519 3/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
LYN P07948 2/20 0.43
BLK P51451 2/20 0.43
DAPK3 O43293 1/20 0.43
RIPK2 O43353 1/20 0.43
EGFR P00533 1/20 0.43
YES1 P07947 1/20 0.43
HCK P08631 1/20 0.43
PDGFRB P09619 1/20 0.43
FGR P09769 1/20 0.43
PDGFRA P16234 1/20 0.43
PRKACA P17612 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162800 0.74 CYP1A2 (0.41) KDRSRCLCKTEKFYN
SCHEMBL30355044 0.74 CYP1A2 (0.41) KDRSRCLCKTEKFYN
SCHEMBL20162797 0.70 CYP1A2 (0.40) KDRSRCLCKTEKFYN
SCHEMBL13020205 0.68 CYP1A2 (0.47) KDRSRCLCKTEKFYN
SCHEMBL20162699 0.67 SRC (0.48) KDRSRCLCKTEKFYN
SCHEMBL20162990 0.67 FYN (0.41) KDRSRCLCKTEKFYN
SCHEMBL30892140 0.66 CFTR (0.51) KDRSRCLCKTEKFYN
SCHEMBL7834490 0.65 EGFR (0.56) KDRSRCLCKTEKABL1
SCHEMBL15708850 0.65 ADK (0.53) KDRSRCLCKTEKFYN
SCHEMBL4065290 0.64 ADK (0.54) KDRSRCABL1ADK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed