SCHEMBL20182299

SCHEMBL20182299

CC(C)(/C(=C/Nc1ccccc1F)N=N)n1cc(-c2ccc(Cl)cc2)c2c(N)ncnc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 10/20 0.54
LCK P06239 7/20 0.54
KDR P35968 7/20 0.54
TEK Q02763 6/20 0.54
BTK Q06187 7/20 0.39
EIF2AK3 Q9NZJ5 3/20 0.38
EGFR P00533 3/20 0.37
ABL1 P00519 2/20 0.37
ABL2 P42684 1/20 0.37
DAPK3 O43293 1/20 0.37
RIPK2 O43353 1/20 0.37
CYP1A2 P05177 1/20 0.37
FYN P06241 1/20 0.37
YES1 P07947 1/20 0.37
LYN P07948 1/20 0.37
HCK P08631 1/20 0.37
PDGFRB P09619 1/20 0.37
FGR P09769 1/20 0.37
CYP2C9 P11712 1/20 0.37
PDGFRA P16234 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20181912 0.78 SRC (0.41) SRCLCKKDRTEKBTK
SCHEMBL3787827 0.72 KDR (1.00) SRCLCKKDRTEKBTK
SCHEMBL20181900 0.70 KDR (0.37) SRCLCKKDRTEKBTK
SCHEMBL20182360 0.70 FYN (0.35) SRCLCKKDRTEKBTK
SCHEMBL20162613 0.70 KDR (0.59) SRCLCKKDRTEKBTK
SCHEMBL30036829 0.70 KDR (0.59) SRCLCKKDRTEKBTK
SCHEMBL20182362 0.69 CFTR (0.40) SRCLCKKDRTEKEGFR
SCHEMBL20182228 0.68 KDR (0.45) SRCLCKKDRTEKBTK
SCHEMBL7010062 0.67 LCK (0.63) SRCLCKKDRTEKBTK
SCHEMBL20182197 0.67 CFTR (0.43) SRCLCKKDRTEKEIF2AK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed