SCHEMBL20182345

SCHEMBL20182345

Cc1nc(N)c2c(C)cn(Cc3cn(-c4ccccc4F)nn3)c2n1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.48
ADORA1 P30542 1/20 0.46
HSP90AA1 P07900 1/20 0.41
PTGS2 P35354 2/20 0.40
PTGS1 P23219 1/20 0.40
RXRA P19793 8/20 0.40
GRIN1 Q05586 7/20 0.40
GRIN2B Q13224 7/20 0.40
CFTR P13569 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
PARP1 P09874 1/20 0.39
GSK3B P49841 1/20 0.36
KCNH2 Q12809 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30038075 0.90 NOTUM (0.46) NOTUMADORA1HSP90AA1PTGS2PTGS1
SCHEMBL20162828 0.90 NOTUM (0.46) NOTUMADORA1HSP90AA1PTGS2PTGS1
SCHEMBL20182215 0.85 NOTUM (0.48) NOTUMHSP90AA1PTGS2PTGS1RXRA
SCHEMBL20162882 0.81 NOTUM (0.39) NOTUMADORA1HSP90AA1RXRAGRIN1
SCHEMBL20162810 0.80 CFTR (0.49) NOTUMADORA1HSP90AA1RXRAGRIN1
SCHEMBL20182201 0.77 NOTUM (0.48) NOTUMHSP90AA1PTGS2PTGS1RXRA
SCHEMBL20162731 0.72 NOTUM (0.48) NOTUMHSP90AA1PTGS2PTGS1RXRA
SCHEMBL20173309 0.72 NOTUM (0.48) NOTUMHSP90AA1PTGS2PTGS1RXRA
SCHEMBL30036886 0.72 NOTUM (0.48) NOTUMHSP90AA1PTGS2PTGS1RXRA
SCHEMBL20163000 0.70 NOTUM (0.46) NOTUMHSP90AA1PTGS2PTGS1RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed