SCHEMBL20182201

SCHEMBL20182201

Cc1cn(Cc2cn(-c3ccccc3F)nn2)c2ncnc(Cl)c12

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.48
PTGS2 P35354 2/20 0.46
RXRA P19793 11/20 0.42
GRIN1 Q05586 10/20 0.42
GRIN2B Q13224 10/20 0.42
HSP90AA1 P07900 1/20 0.41
CFTR P13569 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
PARP1 P09874 1/20 0.39
KCNH2 Q12809 2/20 0.39
PTGS1 P23219 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182215 0.87 NOTUM (0.48) NOTUMPTGS2RXRAGRIN1GRIN2B
SCHEMBL30892138 0.87 NOTUM (0.48) NOTUMPTGS2RXRAGRIN1GRIN2B
SCHEMBL20162698 0.87 NOTUM (0.48) NOTUMPTGS2RXRAGRIN1GRIN2B
SCHEMBL30355045 0.83 PTGS2 (0.42) NOTUMPTGS2RXRAGRIN1GRIN2B
SCHEMBL20163002 0.83 PTGS2 (0.42) NOTUMPTGS2RXRAGRIN1GRIN2B
SCHEMBL20182174 0.81 DRD2 (0.40) GRIN2BCFTRKCNH2
SCHEMBL20173309 0.77 NOTUM (0.48) NOTUMPTGS2RXRAGRIN1GRIN2B
SCHEMBL30036886 0.77 NOTUM (0.48) NOTUMPTGS2RXRAGRIN1GRIN2B
SCHEMBL20182345 0.77 NOTUM (0.48) NOTUMPTGS2RXRAGRIN1GRIN2B
SCHEMBL20162731 0.77 NOTUM (0.48) NOTUMPTGS2RXRAGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed