SCHEMBL20182349

SCHEMBL20182349

CN/C=N/c1ncnc2c1c(I)cn2Cc1cn(-c2ccccc2F)nn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.41
PTGS2 P35354 2/20 0.36
HSP90AA1 P07900 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
PARP1 P09874 1/20 0.34
PDE5A O76074 1/20 0.34
PDE4A P27815 1/20 0.34
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE1C Q14123 1/20 0.34
PDE3A Q14432 1/20 0.34
CFTR P13569 3/20 0.34
CA2 P00918 1/20 0.34
CA5A P35218 1/20 0.34
CA9 Q16790 1/20 0.34
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162823 0.88 NOTUM (0.41) NOTUMPTGS2HSP90AA1TRPV1PARP1
SCHEMBL20162822 0.88 NOTUM (0.41) NOTUMPTGS2HSP90AA1TRPV1PARP1
SCHEMBL20162731 0.80 NOTUM (0.48) NOTUMPTGS2HSP90AA1TRPV1PARP1
SCHEMBL30036886 0.80 NOTUM (0.48) NOTUMPTGS2HSP90AA1TRPV1PARP1
SCHEMBL20162698 0.80 NOTUM (0.48) NOTUMPTGS2HSP90AA1TRPV1PARP1
SCHEMBL30892138 0.80 NOTUM (0.48) NOTUMPTGS2HSP90AA1TRPV1PARP1
SCHEMBL20182201 0.72 NOTUM (0.48) NOTUMPTGS2HSP90AA1TRPV1PARP1
SCHEMBL20182215 0.72 NOTUM (0.48) NOTUMPTGS2HSP90AA1TRPV1PARP1
SCHEMBL20163120 0.72 CFTR (0.44) NOTUMPTGS2HSP90AA1CFTRAMY1A
SCHEMBL20163119 0.72 CFTR (0.44) NOTUMPTGS2HSP90AA1CFTRAMY1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed