SCHEMBL20182356

SCHEMBL20182356

CCC(/C(=C/Nc1ccc(F)cc1F)N=N)n1c(Br)c(-c2cnc(C(F)(F)F)nc2)c2c(N)ncnc21

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CFTR P13569 15/20 0.39
NTRK1 P04629 1/20 0.34
NTRK3 Q16288 1/20 0.34
NTRK2 Q16620 1/20 0.34
RIPK1 Q13546 1/20 0.34
NEK7 Q8TDX7 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182354 0.93 CFTR (0.41) CFTRRIPK1
SCHEMBL20182278 0.91 CFTR (0.37) CFTRNTRK1NTRK3NTRK2RIPK1
SCHEMBL20181896 0.91 CFTR (0.42) CFTRNTRK1NTRK3NTRK2RIPK1
SCHEMBL20182355 0.90 CFTR (0.38) CFTRRIPK1
SCHEMBL20182294 0.85 CFTR (0.40) CFTRNTRK1NTRK3NTRK2RIPK1
SCHEMBL20182263 0.83 CFTR (0.40) CFTRRIPK1
SCHEMBL20182280 0.83 CFTR (0.38) CFTRRIPK1
SCHEMBL20182269 0.81 CFTR (0.38) CFTRRIPK1
SCHEMBL20182268 0.80 CFTR (0.42) CFTRNTRK1NTRK3NTRK2RIPK1
SCHEMBL20181910 0.79 CFTR (0.38) CFTRNTRK1NTRK3NTRK2NEK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed