SCHEMBL20188047

SCHEMBL20188047

C=CCCS(=O)(=O)NC1(c2ccc(F)c(OCC3CCCC3)c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 9/20 0.39
SCN5A Q14524 2/20 0.38
DUT P33316 6/20 0.38
FABP4 P15090 1/20 0.35
FABP5 Q01469 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20188365 0.98 DUT (0.38) SCN9ASCN5ADUT
SCHEMBL20187879 0.97 DUT (0.41) SCN9ADUT
SCHEMBL20377845 0.91 DUT (0.41) DUT
SCHEMBL20351440 0.88 DUT (0.42) SCN9ASCN5ADUTALDH1A1LMNA
SCHEMBL20374175 0.87 DUT (0.44) SCN9ASCN5ADUTALDH1A1LMNA
SCHEMBL20377769 0.86 DUT (0.38) SCN9ADUT
SCHEMBL20351617 0.86 DUT (0.42) SCN9ASCN5ADUT
SCHEMBL20351403 0.85 DUT (0.44) SCN9ASCN5ADUTALDH1A1LMNA
SCHEMBL20351596 0.85 DUT (0.45) SCN9ADUT
SCHEMBL20372976 0.84 DUT (0.46) SCN9ADUT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250188039-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2025-06-12 US disclosed
EP-3319939-B1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS NI LTD (GB) 2024-11-27 EP disclosed
US-12098133-B2 Hydantoin containing deoxyuridine triphosphatase inhibitors CV6 THERAPEUTICS (NI) LIMITED (GB) 2024-09-24 US disclosed
US-20230126280-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2023-04-27 US disclosed
US-11584723-B2 Hydantoin containing deoxyuridine triphosphatase inhibitors CV6 THERAPEUTICS (NI) LIMITED (GB) 2023-02-21 US disclosed
US-20220402879-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2022-12-22 US disclosed
US-11518746-B2 Nitrogen ring linked deoxyuridine triphosphatase inhibitors CV6 THERAPEUTICS (NI) LIMITED (GB) 2022-12-06 US disclosed
US-11247984-B2 Uracil containing compounds CV6 THERAPEUTICS (NI) LIMITED (GB) 2022-02-15 US disclosed
US-11174271-B2 6-membered uracil isosteres CV6 THERAPEUTICS (NI) LIMITED (GB) 2021-11-16 US disclosed
US-11124485-B2 Deoxyuridine triphosphatase inhibitors containing cyclopropano linkage CV6 THERAPEUTICS (NI) LIMITED (GB) 2021-09-21 US disclosed
US-20200039966-A1 URACIL CONTAINING COMPOUNDS CV6 THERAPEUTICS (NI) LIMITED (GB) 2020-02-06 US disclosed
US-10544105-B2 Deoxyuridine triphosphatase inhibitors containing cyclopropano linkage CV6 THERAPEUTICS (NI) LIMITED (GB) 2020-01-28 US disclosed
US-20190330210-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2019-10-31 US disclosed
US-20190276410-A1 NITROGEN RING LINKED DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2019-09-12 US disclosed
US-20190270756-A1 6-MEMBERED URACIL ISOSTERES CV6 THERAPEUTICS (NI) LIMITED (GB) 2019-09-05 US disclosed
US-20180201586-A1 DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CONTAINING CYCLOPROPANO LINKAGE SAI LIFE SCIENCES LIMITED (IN) 2018-07-19 US disclosed
WO-2018128720-A1 URACIL CONTAINING COMPOUNDS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-12 WO disclosed
US-20180194736-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-12 US disclosed
US-20180186737-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-05 US disclosed
WO-2018098207-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (17 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180194736-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD SCN9A 4663/4885SCN5A 4412/4885DUT 1/4885
US-11584723-B2 Hydantoin containing deoxyuridine triphosphatase inhibitors DUT, TYMP, DPYD SCN9A 4663/4885SCN5A 4412/4885DUT 1/4885
US-10544105-B2 Deoxyuridine triphosphatase inhibitors containing cyclopropano linkage DPYD, DUT, TYMP SCN9A 4564/4885SCN5A 4231/4885DUT 2/4885
US-11174271-B2 6-membered uracil isosteres UNG, DUT, DPYD SCN9A 4694/4885SCN5A 4661/4885DUT 2/4885
US-20220402879-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD SCN9A 4663/4885SCN5A 4412/4885DUT 1/4885
US-20190330210-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD SCN9A 4663/4885SCN5A 4412/4885DUT 1/4885
US-20250188039-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD SCN9A 4663/4885SCN5A 4412/4885DUT 1/4885
US-20200039966-A1 URACIL CONTAINING COMPOUNDS UNG, DPYD, DUT SCN9A 4584/4885SCN5A 4492/4885DUT 3/4885
US-11518746-B2 Nitrogen ring linked deoxyuridine triphosphatase inhibitors DUT, DPYD, TYMP SCN9A 4441/4885SCN5A 4331/4885DUT 1/4885
US-11124485-B2 Deoxyuridine triphosphatase inhibitors containing cyclopropano linkage DPYD, DUT, TYMP SCN9A 4564/4885SCN5A 4231/4885DUT 2/4885
US-11247984-B2 Uracil containing compounds UNG, DPYD, DUT SCN9A 4584/4885SCN5A 4492/4885DUT 3/4885
US-20180186737-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD SCN9A 4663/4885SCN5A 4412/4885DUT 1/4885
US-12098133-B2 Hydantoin containing deoxyuridine triphosphatase inhibitors DUT, TYMP, DPYD SCN9A 4663/4885SCN5A 4412/4885DUT 1/4885
US-20190276410-A1 NITROGEN RING LINKED DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, DPYD, TYMP SCN9A 4441/4885SCN5A 4331/4885DUT 1/4885
US-20190270756-A1 6-MEMBERED URACIL ISOSTERES UNG, DUT, DPYD SCN9A 4694/4885SCN5A 4661/4885DUT 2/4885
US-20180201586-A1 DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CONTAINING CYCLOPROPANO LINKAGE DUT, DPYD, TYMP SCN9A 4743/4885SCN5A 4546/4885DUT 1/4885
US-20230126280-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD SCN9A 4663/4885SCN5A 4412/4885DUT 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.