SCHEMBL20190707

SCHEMBL20190707

CN(CC(=O)NC(Cc1ccccn1)c1ccccc1)C(=O)COC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.39
PTPRA P18433 1/20 0.38
HDAC6 Q9UBN7 4/20 0.37
HDAC1 Q13547 2/20 0.37
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HRH2 P25021 1/20 0.37
GAA P10253 1/20 0.37
MAOB P27338 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20188027 0.87 GRIN2D (0.42) PTPRAHDAC6HDAC1HRH2GAA
SCHEMBL20188336 0.87 PTPRA (0.39) PTPRAHDAC6HDAC1HRH2GAA
SCHEMBL20188290 0.86 PTPRA (0.42) PTPRAHDAC6HDAC1HRH2GAA
SCHEMBL20188853 0.86 PTPRA (0.38) PTPRAHDAC6HDAC1HRH2GAA
SCHEMBL22457613 0.86 PTPRA (0.38) PTPRAHDAC6HDAC1HRH2GAA
SCHEMBL29735517 0.86 CYP1A2 (0.39) PTPRAHDAC6HDAC1HRH2GAA
SCHEMBL20187735 0.84 PTPRA (0.40) PTPRAHDAC6HDAC1HRH2GAA
SCHEMBL22457577 0.83 CTSS (0.36) PTPRAHDAC6HDAC1TDP1GAA
SCHEMBL20189051 0.83 CTSS (0.36) PTPRAHDAC6HDAC1TDP1GAA
SCHEMBL20188572 0.82 PTPRA (0.39) PTPRAHDAC6HDAC1KDM4EHRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018098344-A1 PRODRUGS OF LANICEMINE AND THEIR METHOD OF USE BIOHAVEN PHARMACEUTICAL HOLDING COMPANY LTD. (US) 2018-05-31 WO disclosed