SCHEMBL20194290

SCHEMBL20194290

N=Cc1cc(C(=O)Nc2ccccc2N)ccc1NCC1CC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 12/20 0.48
HDAC2 Q92769 10/20 0.48
HDAC3 O15379 8/20 0.48
HDAC4 P56524 5/20 0.48
HDAC7 Q8WUI4 5/20 0.48
HDAC10 Q969S8 5/20 0.48
HDAC11 Q96DB2 5/20 0.48
HDAC8 Q9BY41 5/20 0.48
HDAC6 Q9UBN7 5/20 0.48
HDAC9 Q9UKV0 5/20 0.48
HDAC5 Q9UQL6 5/20 0.48
MAPK1 P28482 1/20 0.45
NCOR2 Q9Y618 2/20 0.44
PTGER4 P35408 1/20 0.44
PTGS1 P23219 1/20 0.43
KDM1A O60341 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20194285 0.88 PTGER4 (0.46) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL20194287 0.87 HDAC1 (0.54) HDAC1HDAC2HDAC3HDAC8NCOR2
SCHEMBL20194284 0.82 HDAC1 (0.60) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL20194283 0.78 HDAC1 (0.52) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL20194294 0.76 HDAC1 (0.48) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL4482782 0.76 HDAC1 (0.62) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL20194282 0.74 HDAC1 (0.43) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL17483922 0.71 HDAC3 (0.60) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL30693377 0.71 PTGER4 (0.47) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL977627 0.71 PTGER4 (0.47) HDAC1HDAC2HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970139-B1 HDAC INHIBITORS BIOMARIN PHARM INC (US) 2018-05-30 EP disclosed