SCHEMBL20203098

SCHEMBL20203098

Fc1cc(F)c(-c2nc3ccccc3n2-c2ccccc2)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.53
HTT P42858 1/20 0.53
GRIA1 P42261 1/20 0.51
CACNG8 Q8WXS5 1/20 0.51
CACNG2 Q9Y698 1/20 0.51
RECQL P46063 1/20 0.49
ESR2 Q92731 4/20 0.49
ESR1 P03372 3/20 0.49
PRKACA P17612 1/20 0.48
RPS6KB1 P23443 1/20 0.48
GSK3B P49841 1/20 0.48
ROCK1 Q13464 1/20 0.48
GSR P00390 1/20 0.44
SCN9A Q15858 2/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20203100 0.85 MAPK1 (0.53) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL21578091 0.84 MAPK1 (0.59) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL3868966 0.82 RECQL (0.53) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL27593044 0.81 RECQL (0.52) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL804817 0.79 MAPK1 (0.66) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL21578020 0.79 MAPK1 (0.53) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL6300348 0.78 RECQL (0.62) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL5581280 0.78 GRIA1 (0.78) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL64508 0.77 ESR2 (0.66) MAPK1HTTGRIA1CACNG8CACNG2
SCHEMBL29351258 0.77 ESR2 (0.66) MAPK1HTTGRIA1CACNG8CACNG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10319920-B2 Carbazole derivatives and organic light-emitting diodes by using the same YUAN ZE UNIVERSITY (TW) 2019-06-11 US disclosed
US-20180151808-A1 CARBAZOLE DERIVATIVES AND ORGANIC LIGHT-EMITTING DIODES BY USING THE SAME YUAN ZE UNIVERSITY (TW) 2018-05-31 US disclosed
US-20180151808-A1 CARBAZOLE DERIVATIVES AND ORGANIC LIGHT-EMITTING DIODES BY USING THE SAME YUAN ZE UNIVERSITY (TW) 2018-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10319920-B2 Carbazole derivatives and organic light-emitting diodes by using the same CBR3, FBXL19, CSNK1A1L MAPK1 3208/4885HTT 2983/4885GRIA1 563/4885
US-20180151808-A1 CARBAZOLE DERIVATIVES AND ORGANIC LIGHT-EMITTING DIODES BY USING THE SAME CBR3, FBXL19, CSNK1A1L MAPK1 3208/4885HTT 2983/4885GRIA1 563/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.