SCHEMBL20203315

SCHEMBL20203315

Cc1cncc2ncn(CC3=NC(C)C(=O)O3)c(=O)c12

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 12/20 0.45
SMN1; SMN2 Q16637 1/20 0.33
TP53 P04637 1/20 0.31
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21363618 0.74 TRPA1 (0.47) TRPA1
SCHEMBL20187600 0.71 TRPA1 (0.52) TRPA1SMN1; SMN2
SCHEMBL20187460 0.67 SMN1; SMN2 (0.45) TRPA1SMN1; SMN2
SCHEMBL22210019 0.66 TRPA1 (0.72) TRPA1
Hydrochloric Acid SCHEMBL22194465 0.65 TRPA1 (0.71) TRPA1
Hydrochloric Acid SCHEMBL22194462 0.65 TRPA1 (0.71) TRPA1
Hydrochloric Acid SCHEMBL22194464 0.65 TRPA1 (0.71) TRPA1
SCHEMBL22210437 0.64 TRPA1 (0.77) TRPA1
SCHEMBL21363471 0.63 TRPA1 (0.37) TRPA1ALDH1A1LMNA
SCHEMBL22477750 0.63 GSK3A (0.39) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096159-A1 OXADIAZOLONES AS TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2018-05-31 WO disclosed