SCHEMBL20203643

SCHEMBL20203643

CC(C)c1ccc2c(n1)CCN(C(=O)C1CN(C)C1)C2

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 10/20 0.40
GRM5 P41594 1/20 0.40
HSP90B1 P14625 4/20 0.39
CDK4 P11802 4/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNE1 P24864 1/20 0.39
GABRG2 P18507 4/20 0.38
GABRB3 P28472 4/20 0.38
GABRA5 P31644 4/20 0.38
KCNH2 Q12809 2/20 0.38
KEAP1 Q14145 1/20 0.37
CDK2 P24941 3/20 0.37
CDK6 Q00534 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20203598 0.92 GRM5 (0.47) HSP90AA1GRM5CDK4CDK1CCNB1
SCHEMBL20203597 0.92 GRM5 (0.47) HSP90AA1GRM5CDK4CDK1CCNB1
SCHEMBL20203457 0.91 GRM5 (0.49) HSP90AA1GRM5CDK4CDK1CCNB1
SCHEMBL22876917 0.85 CDK4 (0.39) HSP90AA1GRM5CDK4CDK1CCNB1
SCHEMBL23733484 0.84 GRM5 (0.42) GRM5CDK4CDK1CCNB1CCNE1
SCHEMBL20203431 0.84 KEAP1 (0.41) HSP90AA1GRM5HSP90B1CDK4CDK1
SCHEMBL23733483 0.83 CDK4 (0.35) HSP90AA1HSP90B1CDK4CDK1GABRG2
SCHEMBL20203456 0.82 GRM5 (0.41) HSP90AA1GRM5CDK4CDK1CCNB1
SCHEMBL20203531 0.82 TLR9 (0.41) HSP90AA1GRM5HSP90B1CDK4CDK1
SCHEMBL21414436 0.82 GRM5 (0.44) HSP90AA1GRM5CDK4CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11084814-B2 Pyrido[3, 4-d]pyrimidine derivative and pharmaceutically acceptable salt thereof TEIJIN PHARMA LIMITED (JP) 2021-08-10 US disclosed
WO-2018097297-A1 PYRIDO[3, 4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 帝人ファーマ株式会社 2018-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11084814-B2 Pyrido[3, 4-d]pyrimidine derivative and pharmaceutically acceptable salt thereof CDK4, CDK6, CDK16 HSP90AA1 4289/4885GRM5 2518/4885HSP90B1 3570/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.