SCHEMBL20203837

SCHEMBL20203837

FC(F)(F)Oc1ccc(-c2cn3c(CC4CCCCO4)nnc3cn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 0.43
SCN5A Q14524 7/20 0.38
SCN1A P35498 1/20 0.38
SCN2A Q99250 1/20 0.38
GLS O94925 1/20 0.36
PIK3CB P42338 1/20 0.35
PRKDC P78527 1/20 0.35
ATM Q13315 1/20 0.35
ATR Q13535 1/20 0.35
ATRIP Q8WXE1 1/20 0.35
TNF P01375 1/20 0.35
USP30 Q70CQ3 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20190811 1.00 CYP1A2 (0.43) CYP1A2SCN5ASCN1ASCN2AGLS
SCHEMBL20190944 1.00 CYP1A2 (0.43) CYP1A2SCN5ASCN1ASCN2AGLS
SCHEMBL20203979 0.82 CYP1A2 (0.42) CYP1A2SCN5ASCN1ASCN2AGLS
SCHEMBL20190711 0.82 CYP1A2 (0.42) CYP1A2SCN5ASCN1ASCN2AGLS
SCHEMBL20190491 0.82 CYP1A2 (0.42) CYP1A2SCN5ASCN1ASCN2AGLS
SCHEMBL20190512 0.81 CYP1A2 (0.61) CYP1A2SCN5ASCN1ASCN2ATNF
SCHEMBL20190661 0.81 CYP1A2 (0.61) CYP1A2SCN5ASCN1ASCN2ATNF
SCHEMBL20203861 0.81 CYP1A2 (0.61) CYP1A2SCN5ASCN1ASCN2ATNF
SCHEMBL20203928 0.78 CYP1A2 (0.62) CYP1A2SCN5ASCN1ASCN2ATNF
SCHEMBL20203803 0.77 CYP1A2 (0.60) CYP1A2SCN5ASCN1ASCN2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018098499-A1 COMPOUNDS AND THEIR METHODS OF USE PRAXIS PRECISION MEDICINES, INC. (US) 2018-05-31 WO disclosed