SCHEMBL20204802

SCHEMBL20204802

C=CC(=O)N1CCc2ccc(C)cc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.51
BTK Q06187 4/20 0.50
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
XIAP P98170 1/20 0.48
BIRC2 Q13490 1/20 0.48
JAK3 P52333 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 4/20 0.43
EGFR P00533 1/20 0.43
FGFR4 P22455 1/20 0.43
CCNK O75909 1/20 0.43
CDK12 Q9NYV4 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.42
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26032620 0.91 ALDH1A1 (0.51) NOTUMBTKSMN1; SMN2KMT2AALDH1A1
SCHEMBL16123336 0.82 BRD4 (0.51) NOTUMBTKJAK3ALDH1A1EGFR
SCHEMBL29782485 0.82 XIAP (0.47) NOTUMBTKXIAPBIRC2ALDH1A1
SCHEMBL17699740 0.82 XIAP (0.47) NOTUMBTKXIAPBIRC2ALDH1A1
SCHEMBL429841 0.81 NOTUM (0.76) NOTUMDRD2DRD4XIAPBIRC2
SCHEMBL31561911 0.81 BTK (0.49) NOTUMBTKJAK3HPGDALDH1A1
SCHEMBL30697880 0.80 MAP2K7 (0.50) BTKJAK3EGFRFGFR4
SCHEMBL27341151 0.80 MAP2K7 (0.50) BTKJAK3EGFRFGFR4
SCHEMBL26691238 0.80 NOTUM (0.55) NOTUMDRD2DRD4XIAPBIRC2
SCHEMBL31562048 0.79 XIAP (0.53) NOTUMBTKXIAPBIRC2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018098473-A1 REAGENTS AND METHODS FOR ANALYSIS OF PROTEINS AND METABOLITES TARGETED BY COVALENT PROBES DANA-FARBER CANCER INSTITUTE, INC. (US) 2018-05-31 WO disclosed