SCHEMBL20209260

SCHEMBL20209260

C[C@H](Nc1nccc(N2CCC[C@H]2CNC(=O)c2ccccc2)n1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 17/20 0.48
MAPK14 Q16539 2/20 0.47
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
CTSK P43235 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20209330 0.86 IDH1 (0.51) IDH1
SCHEMBL30123272 0.85 IDH1 (0.52) IDH1
SCHEMBL30122768 0.85 IDH1 (0.52) IDH1
SCHEMBL20209264 0.85 IDH1 (0.52) IDH1
SCHEMBL20209434 0.83 IDH1 (0.52) IDH1
SCHEMBL20209174 0.83 IDH1 (0.52) IDH1
SCHEMBL20209684 0.81 IDH1 (0.50) IDH1
SCHEMBL20209255 0.81 IDH1 (0.50) IDH1
SCHEMBL20191155 0.78 IDH1 (0.50) IDH1
SCHEMBL20209254 0.78 IDH1 (0.50) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110023298-B Isocitrate Dehydrogenase (IDH) inhibitors 浙江迈同生物医药有限公司 2022-12-16 CN disclosed
WO-2018095344-A1 ISOCITRATE DEHYDROGENASE (IDH) INHIBITOR SHANGHAI METON PHARMACEUTICAL CO., LTD (CN) 2018-05-31 WO disclosed