SCHEMBL20215280

SCHEMBL20215280

Cc1ccccc1Cn1cc(Br)c(=O)nc1-c1cccc(C(F)(F)F)c1Cl

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 18/20 0.55
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20215285 0.91 P2RX7 (0.57) P2RX7KDM4EALDH1A1GAAATM
SCHEMBL20215286 0.89 P2RX7 (0.55) P2RX7KDM4EALDH1A1GAAATM
SCHEMBL20215277 0.86 P2RX7 (0.71) P2RX7
SCHEMBL20215354 0.85 P2RX7 (0.52) P2RX7KDM4EALDH1A1GAAATM
SCHEMBL20215355 0.84 P2RX7 (0.59) P2RX7
SCHEMBL20215352 0.82 P2RX7 (0.56) P2RX7
SCHEMBL20216065 0.80 P2RX7 (0.54) P2RX7
SCHEMBL20215304 0.80 P2RX7 (0.51) P2RX7
SCHEMBL20215362 0.80 P2RX7 (0.62) P2RX7
SCHEMBL20215350 0.79 P2RX7 (0.61) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed