SCHEMBL20217299

SCHEMBL20217299

N=C(c1ccc(PCCN2CCOCC2)cc1)c1cc(C(=O)NC(c2ccccc2)C2CC2)ccc1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 5/20 0.37
HDAC3 O15379 4/20 0.37
HDAC1 Q13547 4/20 0.37
KCNK3 O14649 1/20 0.37
F10 P00742 3/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
F2 P00734 2/20 0.35
PRSS1 P07477 2/20 0.35
ROCK2 O75116 2/20 0.35
AKT1 P31749 2/20 0.35
SMYD3 Q9H7B4 1/20 0.35
CDK2 P24941 1/20 0.35
ROCK1 Q13464 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217295 0.86 SMN1; SMN2 (0.47) HDAC1MEN1ALDH1A1KMT2A
SCHEMBL20217236 0.84 HDAC3 (0.44) HDAC2HDAC3HDAC1KCNK3F10
SCHEMBL20217262 0.81 F10 (0.46) HDAC2HDAC3HDAC1KCNK3F10
SCHEMBL20217694 0.79 MEN1 (0.47) F10MEN1ALDH1A1MAPK1KMT2A
SCHEMBL20217743 0.78 MEN1 (0.45) F10MEN1ALDH1A1MAPK1KMT2A
SCHEMBL20217335 0.78 F10 (0.43) KCNK3F10MEN1ALDH1A1MAPK1
SCHEMBL20217296 0.77 TTK (0.50) F10MEN1ALDH1A1MAPK1KMT2A
SCHEMBL20217747 0.77 CYP3A4 (0.47) KCNK3F10MEN1ALDH1A1MAPK1
SCHEMBL20217712 0.76 F10 (0.44) KCNK3F10MEN1ALDH1A1MAPK1
SCHEMBL20217185 0.76 AKT1 (0.43) HDAC2HDAC3HDAC1KCNK3F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed