SCHEMBL20217296

SCHEMBL20217296

N=C(c1ccc(OC2CCN(CCF)CC2)cc1)c1cc(C(=O)NC(c2ccccc2)C2CC2)ccc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 5/20 0.50
CYP3A4 P08684 4/20 0.50
AURKB Q96GD4 3/20 0.47
INCENP Q9NQS7 3/20 0.47
LMNA P02545 4/20 0.42
ALDH1A1 P00352 3/20 0.42
SLC5A7 Q9GZV3 2/20 0.42
PKM P14618 1/20 0.42
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
MAPK1 P28482 1/20 0.40
SRD5A1 P18405 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
AKT1 P31749 2/20 0.37
CDK2 P24941 1/20 0.37
F10 P00742 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217221 0.90 TTK (0.51) TTKCYP3A4AURKBINCENPLMNA
SCHEMBL20217268 0.89 MEN1 (0.47) TTKCYP3A4AURKBINCENPLMNA
SCHEMBL20217198 0.87 CYP3A4 (0.52) TTKCYP3A4AURKBINCENPLMNA
SCHEMBL20217290 0.86 ALDH1A1 (0.49) TTKCYP3A4AURKBINCENPLMNA
SCHEMBL20217747 0.84 CYP3A4 (0.47) TTKCYP3A4AURKBINCENPLMNA
SCHEMBL20217390 0.84 TTK (0.63) TTKCYP3A4AURKBINCENPLMNA
SCHEMBL20217292 0.82 TTK (0.39) TTKCYP3A4AURKBINCENPLMNA
SCHEMBL20217295 0.81 SMN1; SMN2 (0.47) LMNAALDH1A1MEN1KMT2ARAB9A
SCHEMBL20217409 0.81 LMNA (0.44) TTKCYP3A4LMNAALDH1A1SLC5A7
SCHEMBL20217694 0.81 MEN1 (0.47) TTKCYP3A4AURKBINCENPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed