SCHEMBL20233293

SCHEMBL20233293

O=C(NNS(=O)(=O)c1ccccc1)c1ccc(Cl)cc1

nearest known ligand 0.78

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 8/20 0.78
MEN1 O00255 2/20 0.77
KMT2A Q03164 2/20 0.77
GAA P10253 4/20 0.68
HTT P42858 1/20 0.67
FLT1 P17948 2/20 0.62
FLT4 P35916 2/20 0.62
KDR P35968 2/20 0.62
L3MBTL1 Q9Y468 1/20 0.62
ALDH1A1 P00352 1/20 0.61
BCAT1 P54687 1/20 0.61
CYP3A4 P08684 1/20 0.58
PKM P14618 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765513 0.88 KAT6A (1.00) KAT6AMEN1KMT2AGAAHTT
SCHEMBL26104327 0.87 MEN1 (1.00) KAT6AMEN1KMT2AGAAHTT
SCHEMBL6400145 0.85 KAT6A (0.81) KAT6AMEN1KMT2AGAAHTT
SCHEMBL20233361 0.84 KAT6A (0.78) KAT6AMEN1KMT2AGAAHTT
SCHEMBL6396355 0.84 KAT6A (0.78) KAT6AMEN1KMT2AGAAHTT
SCHEMBL20465469 0.83 KAT6A (1.00) KAT6AGAA
SCHEMBL20233371 0.83 KAT6A (0.85) KAT6AGAA
SCHEMBL15047783 0.82 KAT6A (0.60) KAT6AMEN1KMT2AGAAFLT1
SCHEMBL6397060 0.81 KAT6A (0.73) KAT6AMEN1KMT2AGAAHTT
SCHEMBL6979280 0.81 KAT6A (0.73) KAT6AMEN1KMT2AGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018102419-A1 COMPOUNDS CONTAINING A SULFONIC GROUP AS KAT INHIBITORS Epizyme, Inc. (US) 2018-06-07 WO disclosed