SCHEMBL20243776

SCHEMBL20243776

N#Cc1ccccc1/C=C/C=C1C(=O)NC(O)NC1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 2/20 0.36
F2R P25116 2/20 0.35
DOCK2 Q92608 1/20 0.34
MAPT P10636 3/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPK1 P28482 2/20 0.32
KMT2A Q03164 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
HTT P42858 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
NTSR1 P30989 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SOS1 Q07889 1/20 0.31
MCL1 Q07820 1/20 0.31
APP P05067 1/20 0.31
SNCA P37840 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14712955 0.82 METAP1 (0.56) METAP1F2RDOCK2MAPTKDM4E
SCHEMBL19820143 0.75 HDAC2 (0.42) METAP1MAPTKDM4EALDH1A1MAPK1
SCHEMBL14713024 0.73 MAPT (0.45) METAP1DOCK2MAPTKDM4EALDH1A1
SCHEMBL5561570 0.69 CDK4 (0.52) F2RMAPTKDM4EALDH1A1MAPK1
SCHEMBL628777 0.69 CDK4 (0.52) F2RMAPTKDM4EALDH1A1MAPK1
SCHEMBL7905215 0.68 TSHR (0.48) F2RKDM4EALDH1A1HTTLMNA
SCHEMBL29732385 0.68 TSHR (0.48) F2RKDM4EALDH1A1HTTLMNA
SCHEMBL1932223 0.68 TSHR (0.48) F2RKDM4EALDH1A1HTTLMNA
SCHEMBL9187108 0.66 TSHR (0.46) F2RKDM4EALDH1A1HTTLMNA
SCHEMBL1399132 0.66 CA1 (0.43) F2RMAPTKDM4EALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9994554-B2 Barbiturate and thiobarbiturate compounds for use in cancer therapy NUHOPE LLC (US) 2018-06-12 US disclosed