SCHEMBL29732385

SCHEMBL29732385

N#Cc1ccccc1C=Cc1ccccc1C#N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.48
NFE2L2 Q16236 1/20 0.40
F2R P25116 3/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ESR2 Q92731 1/20 0.39
IMPDH2 P12268 2/20 0.38
IMPDH1 P20839 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MCL1 Q07820 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HTT P42858 2/20 0.36
ALDH1A1 P00352 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7905215 1.00 TSHR (0.48) TSHRNFE2L2F2RCA1CA2
SCHEMBL1932223 1.00 TSHR (0.48) TSHRNFE2L2F2RCA1CA2
SCHEMBL9187108 0.97 TSHR (0.46) TSHRNFE2L2F2RCA1CA2
SCHEMBL553823 0.91 NR1H3 (0.44) TSHRNFE2L2CYP1A2LMNA
SCHEMBL21574808 0.91 NR1H3 (0.44) TSHRNFE2L2CYP1A2LMNA
SCHEMBL29392092 0.91 NR1H3 (0.44) TSHRNFE2L2CYP1A2LMNA
SCHEMBL553822 0.91 NR1H3 (0.44) TSHRNFE2L2CYP1A2LMNA
SCHEMBL1674897 0.89 NFE2L2 (0.50) TSHRNFE2L2ALDH1A1HPGD
Benzene SCHEMBL29196105 0.89 NFE2L2 (0.50) TSHRNFE2L2ALDH1A1HPGD
SCHEMBL29628296 0.89 NFE2L2 (0.50) TSHRNFE2L2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4232014-A1 ANALOGUES OF PENTAMIDINE AND METHODS FOR TREATING INFECTIONS Auransa Inc. (US) 2023-08-30 EP disclosed
WO-2022087636-A1 ANALOGUES OF PENTAMIDINE AND METHODS FOR TREATING INFECTIONS AURANSA INC. (US) 2022-04-28 WO disclosed