SCHEMBL20247403

SCHEMBL20247403

CCCOc1cc(C(=O)OCC)cc(C)c1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.47
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA7 P43166 3/20 0.46
CA9 Q16790 3/20 0.46
CA14 Q9ULX7 3/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B2 P37059 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 1/20 0.41
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAOA P21397 1/20 0.40
CYP2C19 P33261 1/20 0.40
SCN1A P35498 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16055171 0.90 MEN1 (0.51) ESR1CA12CA1CA2CA7
SCHEMBL16055776 0.87 CA12 (0.49) ESR1CA12CA1CA2CA7
SCHEMBL24408044 0.84 KDM4E (0.51) ESR1CA12CA1CA2CA7
SCHEMBL1425609 0.84 ESR1 (0.41) ESR1CA12CA1CA2CA7
SCHEMBL25276513 0.82 CA12 (0.60) ESR1CA12CA1CA2CA7
SCHEMBL7930568 0.81 CA12 (0.51) ESR1CA12CA1CA2CA7
SCHEMBL28201667 0.81 CA12 (0.51) CA12CA1CA2CA7CA9
SCHEMBL289285 0.81 CA12 (0.55) ESR1CA12CA1CA2CA7
SCHEMBL7930563 0.80 CA12 (0.50) ESR1CA12CA1CA2CA7
SCHEMBL7730273 0.80 ESR1 (0.56) ESR1CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3055309-B1 ANTAGONISTS OF SOMATOSTATIN RECEPTOR SUBTYPE 5 (SSTR5) TAKEDA PHARMACEUTICALS CO (JP) 2018-06-13 EP disclosed