SCHEMBL20249140

SCHEMBL20249140

CC(C)(C)c1ccc(CN2CCNC3(CC3)C2)cn1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.38
MGLL Q99685 1/20 0.35
CCR9 P51686 3/20 0.35
PPARD Q03181 1/20 0.35
MOGAT2 Q3SYC2 4/20 0.33
RET P07949 1/20 0.33
PDCD1LG2 Q9BQ51 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
KDM1A O60341 1/20 0.32
MAOB P27338 1/20 0.32
RCOR1 Q9UKL0 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20249139 0.86 IDH1 (0.37) IDH1MGLLCCR9PPARDMOGAT2
SCHEMBL20038218 0.83 IDH1 (0.39) IDH1PDCD1LG2CD274KDM1AMAOB
SCHEMBL20037913 0.81 IDH1 (0.37) IDH1PDCD1LG2CD274KDM1AMAOB
SCHEMBL18291431 0.81 IDH1 (0.37) IDH1PDCD1LG2CD274CHRNB2CHRNB4
SCHEMBL20224126 0.80 CXCR4 (0.49) PPARD
SCHEMBL20038157 0.79 PRMT5 (0.38) IDH1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL20249346 0.78 PANK3 (0.37) CCR9
SCHEMBL20037439 0.78 IDH1 (0.36) IDH1PDCD1LG2CD274KDM1AMAOB
SCHEMBL20249264 0.75 CXCR4 (0.58)
SCHEMBL12673217 0.75 HRH3 (0.50) PPARDCHRNB2CHRNA4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 IDH1 147/4885MGLL 4576/4885CCR9 2183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.