SCHEMBL20249264

SCHEMBL20249264

CC(C)(C)c1ccc(CN2CCCNCC2)cn1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 15/20 0.58
MEN1 O00255 1/20 0.57
CHRM2 P08172 1/20 0.57
CHRM1 P11229 1/20 0.57
ADRA2C P18825 1/20 0.57
CCR2 P41597 1/20 0.57
CXCL12 P48061 1/20 0.57
BLM P54132 1/20 0.57
KMT2A Q03164 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
HRH3 Q9Y5N1 1/20 0.57
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20224126 0.94 CXCR4 (0.49) CXCR4MEN1CHRM2CHRM1ADRA2C
SCHEMBL12673217 0.87 HRH3 (0.50) TDP1HRH3
SCHEMBL14747471 0.86 HRH3 (0.53) TDP1HRH3
SCHEMBL26351870 0.86 HRH3 (0.53) TDP1HRH3
SCHEMBL22642370 0.83 PARP1 (0.46) CXCR4MEN1CHRM2CHRM1ADRA2C
SCHEMBL20037919 0.82 CXCR4 (0.62) CXCR4MEN1CHRM2CHRM1ADRA2C
SCHEMBL4757141 0.80 PPARD (0.49) CXCR4MEN1CHRM2CHRM1ADRA2C
SCHEMBL20249126 0.79 GRM5 (0.42) KMT2A
SCHEMBL20038107 0.79 CXCR4 (0.62) CXCR4MEN1CHRM2CHRM1ADRA2C
Hydrochloric Acid SCHEMBL27861921 0.79 CXCR4 (0.49) CXCR4MEN1CHRM2CHRM1ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 CXCR4 1021/4885MEN1 2609/4885CHRM2 4833/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.