SCHEMBL20249158

SCHEMBL20249158

CC(C)(C)c1ccc(CN2CC[C@@H](O)C2)cn1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
CD274 Q9NZQ7 3/20 0.43
PDCD1 Q15116 2/20 0.43
LTA4H P09960 9/20 0.42
MEN1 O00255 1/20 0.42
CYP2D6 P10635 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
SPHK1 Q9NYA1 2/20 0.40
SPHK2 Q9NRA0 1/20 0.40
CNR2 P34972 1/20 0.40
KCNH2 Q12809 1/20 0.39
GPR119 Q8TDV5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20249418 1.00 ALDH1A1 (0.47) ALDH1A1KDM4EGAACD274PDCD1
SCHEMBL20249108 0.92 ALDH1A1 (0.55) ALDH1A1KDM4EGAALTA4HCNR2
SCHEMBL20249510 0.92 ALDH1A1 (0.55) ALDH1A1KDM4EGAALTA4HCNR2
SCHEMBL20249506 0.92 ALDH1A1 (0.55) ALDH1A1KDM4EGAALTA4HCNR2
SCHEMBL20249121 0.92 ALDH1A1 (0.52) ALDH1A1KDM4EGAACD274PDCD1
SCHEMBL20249107 0.89 CCR9 (0.41) CD274PDCD1LTA4HMEN1KMT2A
SCHEMBL20249161 0.85 HRH3 (0.45) LTA4HKMT2AKCNH2GPR119
SCHEMBL20249155 0.82 S1PR5 (0.54) CD274PDCD1LTA4HKMT2A
SCHEMBL20249249 0.82 PPARD (0.43) LTA4HKMT2AKCNH2GPR119
SCHEMBL20249125 0.81 HRH3 (0.45) LTA4HKMT2AKCNH2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 ALDH1A1 944/4885KDM4E 470/4885GAA 2747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.