SCHEMBL20249196

SCHEMBL20249196

CN(C)CCOc1ccc(C(C)(C)C)nc1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.53
CHRNA4 P43681 2/20 0.53
HRH3 Q9Y5N1 1/20 0.49
LTA4H P09960 2/20 0.47
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20249212 0.92 KDM4E (0.53) CHRNB2CHRNA4HRH3KDM4E
SCHEMBL25888663 0.81 CA12 (0.47) CHRNB2CHRNA4LTA4H
SCHEMBL20128692 0.81 CA12 (0.47) LTA4HKDM4E
SCHEMBL20249203 0.79 CYP3A4 (0.47) CHRNB2CHRNA4
SCHEMBL22043410 0.79 CBFB (0.40) KDM4E
SCHEMBL25053677 0.78 NR5A1 (0.47) LTA4HKDM4E
SCHEMBL20249214 0.78 CYP3A4 (0.39)
SCHEMBL26796046 0.77 CHRNB2 (0.49) CHRNB2CHRNA4HRH3LTA4HKEAP1
SCHEMBL14308132 0.77 CHRNB2 (0.62) CHRNB2CHRNA4HRH3LTA4HKEAP1
SCHEMBL12710188 0.77 NQO1 (0.50) LTA4HKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 CHRNB2 4863/4885CHRNA4 4628/4885HRH3 2304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.