SCHEMBL4757141

SCHEMBL4757141

FC(F)(F)c1ccc(CN2CCNCC2)cn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 1/20 0.49
CXCR4 P61073 11/20 0.47
MEN1 O00255 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
ADRA2C P18825 1/20 0.47
CCR2 P41597 1/20 0.47
CXCL12 P48061 1/20 0.47
BLM P54132 1/20 0.47
KMT2A Q03164 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
JAK2 O60674 1/20 0.46
JAK1 P23458 1/20 0.46
TYK2 P29597 1/20 0.46
JAK3 P52333 1/20 0.46
KCNH2 Q12809 1/20 0.43
GPR119 Q8TDV5 1/20 0.43
ADRB1 P08588 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27861921 0.98 CXCR4 (0.49) PPARDCXCR4MEN1CHRM2CHRM1
SCHEMBL21607905 0.91 PPARD (0.47) PPARDCXCR4MEN1CHRM2CHRM1
Tert-Butyl Formate SCHEMBL27844698 0.87 PPARD (0.53) PPARDCXCR4MEN1CHRM2CHRM1
SCHEMBL20224126 0.85 CXCR4 (0.49) PPARDCXCR4MEN1CHRM2CHRM1
SCHEMBL28191749 0.84 ALDH1A1 (0.58) PPARDHRH3JAK2JAK1TYK2
SCHEMBL22642370 0.82 PARP1 (0.46) PPARDCXCR4MEN1CHRM2CHRM1
SCHEMBL25145683 0.82 PPARD (0.45) PPARDMEN1KMT2AJAK2JAK1
SCHEMBL18389831 0.82 PPARD (0.55) PPARDJAK2JAK1TYK2JAK3
SCHEMBL20382071 0.82 PPARD (0.55) PPARDMEN1KMT2AJAK2JAK1
SCHEMBL22642373 0.80 HRH3 (0.48) CXCR4MEN1CHRM2CHRM1ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020012424-A1 SUBSTITUTED (AZA)INDOLE DERIVATIVES RICHTER GEDEON NYRT. (HU) 2020-01-16 WO disclosed
WO-2012019430-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-02-16 WO disclosed
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed