SCHEMBL20255151

SCHEMBL20255151

CN1CCN(c2ccc(C(C)(C)CCC(C)(C)c3ccc(N4CCN(CCO)CC4)cn3)nc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.42
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
SYK P43405 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
PARP1 P09874 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
CHKA P35790 1/20 0.38
HRH1 P35367 1/20 0.38
TLR9 Q9NR96 1/20 0.37
CYP3A4 P08684 1/20 0.37
LSS P48449 1/20 0.37
TERT O14746 1/20 0.37
CDK1 P06493 1/20 0.37
CDK4 P11802 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNA2 P20248 1/20 0.37
CCND1 P24385 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20249105 0.85 GAA (0.46) GAAALDH1A1SYKPPARDPPARA
SCHEMBL25160141 0.77 PARP1 (0.47) GAAKDM4EALDH1A1PARP1PARP2
SCHEMBL20085931 0.76 MAPT (0.46) GAAKDM4EALDH1A1MAPTHTR3A
SCHEMBL11981570 0.76 MAPT (0.44) GAAKDM4EALDH1A1HTTHRH1
SCHEMBL20255358 0.75 PPARD (0.42) PPARDPPARAPARP1PARP2MEN1
SCHEMBL17226924 0.73 MAPT (0.42) GAAKDM4EALDH1A1HTTPARP1
SCHEMBL20037559 0.73 GAA (0.43) GAASYKHRH1TLR9CYP3A4
SCHEMBL12595113 0.73 AKR1C3 (0.51) GAAHRH1CDK1CDK4CCNB1
SCHEMBL12595075 0.73 GAA (0.43) GAASYKHRH1TLR9CYP3A4
SCHEMBL20332608 0.73 ROCK2 (0.46) GAAKDM4ESYKHRH1TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 GAA 2747/4885KDM4E 470/4885ALDH1A1 944/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.