SCHEMBL20266409

SCHEMBL20266409

O=C(O)c1ccc2nc(CCl)n(C[C@@H]3CCO3)c2c1

nearest known ligand 0.50

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GLP1R P43220 20/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20266411 1.00 GLP1R (0.50) GLP1R
SCHEMBL27154428 1.00 GLP1R (0.50) GLP1R
SCHEMBL25382123 0.91 GLP1R (0.49) GLP1R
SCHEMBL29668740 0.91 GLP1R (0.49) GLP1R
SCHEMBL25366115 0.91 PTGER4 (0.55) GLP1R
SCHEMBL25366110 0.91 PTGER4 (0.55) GLP1R
SCHEMBL29053103 0.90 GLP1R (0.42) GLP1R
SCHEMBL26482529 0.90 GLP1R (0.49) GLP1R
SCHEMBL27110957 0.90 GLP1R (0.49) GLP1R
SCHEMBL29149774 0.89 GLP1R (0.50) GLP1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 80 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024018395-A1 METHODS AND INTERMEDIATES FOR PREPARING 2-[(4-{6-[(4-CYANO-2-FLUOROBENZYL)OXY]PYRIDIN-2-YL}PIPERIDIN-1-YL)METHYL]-1-[(2S)-OXETAN-2-YLMETHYL]-1H-BENZIMIDAZOLE-6-CARBOXYLIC ACID, 1,3-DIHYDROXY-2-(HYDROXYMETHYL)PROPAN-2-AMINE SALT PFIZER INC. (US) 2024-01-25 WO claimed
US-12595249-B2 Aryl ether-substituted heterocyclic compounds as glpir agonists MINDRANK AI LTD. (CN) 2026-04-07 US disclosed
US-12590081-B2 Fused imidazole derivatives, preparation method and medicinal use thereof JIANGSU HENGRUI PHARMACEUTICALS CO., LTD. (CN) 2026-03-31 US disclosed
US-12497384-B2 Aryl ether-substituted heterocyclic compounds as GLP1R agonists MINDRANK AI LTD. (CN) 2025-12-16 US disclosed
US-20250304553-A1 ARYL ETHER-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS GLP1R AGONISTS MINDRANK AI LTD. (CN) 2025-10-02 US disclosed
US-20250282757-A1 ARYL ETHER-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS GLP1R AGONISTS MINDRANK AI LTD. (CN) 2025-09-11 US disclosed
CN-117242067-B Novel aryl ether substituted heterocycles as GLP1R agonists 杭州德睿智药科技有限公司 2025-03-25 CN disclosed
CN-115594669-B Parallel ring derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2024-11-05 CN disclosed
CN-118420603-A Tromethamine salt crystal form of cycloolefin compound and preparation method and application thereof 江苏豪森药业集团有限公司 2024-08-02 CN disclosed
WO-2024153041-A1 METHOD FOR MANUFACTURING GLP-1R AGONIST, INTERMEDIATE, AND USE THEREOF 杭州德睿智药科技有限公司 2024-07-25 WO disclosed
US-10851081-B2 GLP-1 receptor agonists and uses thereof PFIZER INC. (US) 2020-12-01 US disclosed
US-10844049-B2 GLP-1R agonists and uses thereof QILU REGOR THERAPEUTICS INC. (CN) 2020-11-24 US disclosed
US-20200283424-A1 GLP-1R AGONISTS AND USES THEREOF QILU REGOR THERAPEUTICS INC. (CN) 2020-09-10 US disclosed
US-20200255406-A1 GLP-1 RECEPTOR AGONISTS AND USES THEREOF PFIZER INC. (US) 2020-08-13 US disclosed
US-10669259-B2 GLP-1 receptor agonists and uses thereof PFIZER INC. (US) 2020-06-02 US disclosed
EP-3555064-A1 GLP-1 RECEPTOR AGONISTS AND USES THEREOF Pfizer Inc. (US) 2019-10-23 EP disclosed
US-20190119255-A1 GLP-1 Receptor Agonists and Uses Thereof PFIZER INC. (US) 2019-04-25 US disclosed
US-10208019-B2 GLP-1 receptor agonists and uses thereof PFIZER INC. (US) 2019-02-19 US disclosed
US-20180170908-A1 GLP-1 Agonists and Uses Thereof PFIZER INC. (US) 2018-06-21 US disclosed
WO-2018109607-A1 GLP-1 RECEPTOR AGONISTS AND USES THEREOF PFIZER INC. (US) 2018-06-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10669259-B2 GLP-1 receptor agonists and uses thereof GLP1R, GIPR, GPR119 GLP1R 1/4885
US-12497384-B2 Aryl ether-substituted heterocyclic compounds as GLP1R agonists GLP1R, GIPR, GCGR GLP1R 1/4885
US-12595249-B2 Aryl ether-substituted heterocyclic compounds as glpir agonists GLP1R, GIPR, GCGR GLP1R 1/4885
US-20250304553-A1 ARYL ETHER-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS GLP1R AGONISTS GLP1R, GIPR, GCGR GLP1R 1/4885
US-10844049-B2 GLP-1R agonists and uses thereof GLP1R, GPR119, GIPR GLP1R 1/4885
US-12590081-B2 Fused imidazole derivatives, preparation method and medicinal use thereof GLP1R, GIPR, GPR119 GLP1R 1/4885
US-20180170908-A1 GLP-1 Agonists and Uses Thereof GLP1R, GIPR, GPR119 GLP1R 1/4885
US-20200283424-A1 GLP-1R AGONISTS AND USES THEREOF GLP1R, GPR119, GIPR GLP1R 1/4885
US-10851081-B2 GLP-1 receptor agonists and uses thereof GLP1R, GIPR, GPR119 GLP1R 1/4885
US-20190119255-A1 GLP-1 Receptor Agonists and Uses Thereof GLP1R, GIPR, GPR119 GLP1R 1/4885
US-10208019-B2 GLP-1 receptor agonists and uses thereof GLP1R, GIPR, GPR119 GLP1R 1/4885
US-20250282757-A1 ARYL ETHER-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS GLP1R AGONISTS GLP1R, GIPR, GCGR GLP1R 1/4885
US-20200255406-A1 GLP-1 RECEPTOR AGONISTS AND USES THEREOF GLP1R, GIPR, GPR119 GLP1R 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.