SCHEMBL20280968

SCHEMBL20280968

C[C@H]1CCC[C@H](N2CCOCC2)C1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
TSHR P16473 1/20 0.42
USP2 O75604 1/20 0.36
CYP2A13 Q16696 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
L3MBTL3 Q96JM7 1/20 0.35
OPRL1 P41146 2/20 0.34
SETD2 Q9BYW2 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16907747 1.00 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2TSHRUSP2CYP2A13
SCHEMBL22179798 0.88 SMN1; SMN2 (0.41) ALDH1A1SMN1; SMN2CYP2A13L3MBTL1L3MBTL3
SCHEMBL26820276 0.88 SMN1; SMN2 (0.41) ALDH1A1SMN1; SMN2CYP2A13L3MBTL1L3MBTL3
SCHEMBL26820274 0.88 SMN1; SMN2 (0.41) ALDH1A1SMN1; SMN2CYP2A13L3MBTL1L3MBTL3
SCHEMBL14355430 0.85 ALDH1A1 (0.54) ALDH1A1TSHRUSP2HRH3
SCHEMBL23517478 0.83 ALDH1A1 (0.49) ALDH1A1TSHRUSP2L3MBTL1L3MBTL3
SCHEMBL16566607 0.83 ALDH1A1 (0.49) ALDH1A1TSHRUSP2L3MBTL1L3MBTL3
SCHEMBL15468146 0.81 ALDH1A1 (0.47) ALDH1A1TSHRUSP2L3MBTL1L3MBTL3
SCHEMBL12716769 0.81 CYP2A13 (0.46) ALDH1A1SMN1; SMN2CYP2A13L3MBTL1L3MBTL3
SCHEMBL8378166 0.81 CYP2A13 (0.46) ALDH1A1SMN1; SMN2CYP2A13L3MBTL1L3MBTL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022115879-A1 PYRROLIDINE DERIVATIVES AND METHODS OF USE GENENTECH, INC. (US) 2022-06-02 WO disclosed
US-20180169094-A1 PYRIMIDINE PYRAZOLYL DERIVATIVES AND THEIR USE AS IRAK INHIBITORS MERCK PATENT GMBH (DE) 2018-06-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180169094-A1 PYRIMIDINE PYRAZOLYL DERIVATIVES AND THEIR USE AS IRAK INHIBITORS IRAK2, IRAK3, IRAK1 ALDH1A1 1540/4885SMN1; SMN2 3790/4885TSHR 2324/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.