SCHEMBL20283147

SCHEMBL20283147

CNC1CN(c2ncccc2F)C1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.48
CHRM4 P08173 1/20 0.46
GRM1 Q13255 2/20 0.45
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
CDC42BPB Q9Y5S2 1/20 0.43
HRH3 Q9Y5N1 2/20 0.39
HRH4 Q9H3N8 8/20 0.38
CHI3L1 P36222 1/20 0.38
KCNH2 Q12809 1/20 0.38
CHIT1 Q13231 1/20 0.38
CHI3L2 Q15782 1/20 0.38
CHIA Q9BZP6 1/20 0.38
TRPV1 Q8NER1 1/20 0.37
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23046573 0.83 GRM4 (0.46) GRM4CHRM4GRM1ROCK2ROCK1
SCHEMBL18136223 0.81 GRM1 (0.48) GRM4CHRM4GRM1HRH3CHI3L1
SCHEMBL20283136 0.81 HSD11B1 (0.48) GRM4HRH4KCNH2TRPV1
SCHEMBL18133860 0.77 GRM1 (0.45) GRM4CHRM4GRM1HRH3CHI3L1
SCHEMBL29414908 0.77 GRM1 (0.45) GRM4CHRM4GRM1HRH3CHI3L1
SCHEMBL19116107 0.77 GRM1 (0.45) GRM4CHRM4GRM1HRH3CHI3L1
SCHEMBL19115704 0.77 GRM1 (0.45) GRM4CHRM4GRM1HRH3CHI3L1
SCHEMBL22210095 0.75 GRM1 (0.43) GRM4CHRM4GRM1HRH3CHI3L1
SCHEMBL20283138 0.75 HRH4 (0.40) HRH3HRH4KCNH2
SCHEMBL31595778 0.74 GRM1 (0.48) GRM4CHRM4GRM1HRH3CHI3L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018112312-A1 POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2018-06-21 WO disclosed