SCHEMBL2028830

SCHEMBL2028830

COC(O)C(C)NC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.33
CA14 Q9ULX7 2/20 0.32
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
CA12 O43570 2/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP8 P22894 1/20 0.30
CA9 Q16790 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19477950 0.81 TRPV1 (0.41) CA14CA12CA1CA2MMP1
SCHEMBL15562023 0.79 TP53 (0.32) TP53CA14CYP2D6CYP2C19
SCHEMBL4440551 0.78 POLB (0.40) CYP2D6CYP2C19CA12CA1CA2
SCHEMBL28719441 0.76 CYP2D6 (0.41) TP53CYP2D6CYP2C19CA12CA1
SCHEMBL2026408 0.76 MGAM (0.34) CYP2D6CYP2C19MMP8SMN1; SMN2
SCHEMBL2024610 0.74 SLC1A3 (0.41) CYP2D6CYP2C19
SCHEMBL25170149 0.74 MLYCD (0.30)
SCHEMBL23457853 0.74
SCHEMBL16823439 0.74 TP53 (0.40) TP53CYP2D6CYP2C19
SCHEMBL14952782 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064493-A1 COMPOUNDS AND METHODS FOR TREATING CORONAVIRUSES Clear Creek Bio, Inc. (US) 2023-04-20 WO disclosed
EP-3374359-A1 DIHYDROIMIDAZOPYRAZINONE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Astrazeneca AB (SE) 2018-09-19 EP disclosed
WO-2017080979-A1 DIHYDROIMIDAZOPYRAZINONE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2017-05-18 WO disclosed
WO-2016162325-A1 SUBSTITUTED 3,4-DIHYDROPYRROLO[1,2-A]PYRAZIN-1 (2H)-ONE DERIVATIVES AS KINASE INHIBITORS ASTRAZENECA AB (SE) 2016-10-13 WO disclosed
WO-2014178082-A1 NOVEL 2'/3'/5'-(R/S)-SERINYL FUNCTIONALIZED OLIGONUCLEOTIDES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2014-11-06 WO disclosed
WO-2014022752-A1 MACROCYCLES AS PIM INHIBITORS AMGEN INC. (US) 2014-02-06 WO disclosed
EP-2516434-A1 FUSED HETEROAROMATIC PYRROLIDINONES AS SYK INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2012-10-31 EP disclosed
WO-2011079051-A1 FUSED HETEROAROMATIC PYRROLIDINONES AS SYK INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-06-30 WO disclosed