SCHEMBL20308908

SCHEMBL20308908

COc1cc(C)cc(-c2c(NC(C)c3ccccc3)ccc3ccccc23)c1O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 5/20 0.41
EGFR P00533 5/20 0.41
KRAS P01116 3/20 0.41
MAPT P10636 4/20 0.38
KMT2A Q03164 5/20 0.37
MEN1 O00255 4/20 0.37
HTT P42858 1/20 0.37
HIF1A Q16665 1/20 0.37
STAT3 P40763 1/20 0.36
P4HB P07237 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19672933 1.00 SOS1 (0.41) SOS1EGFRKRASMAPTKMT2A
SCHEMBL19672931 0.83 RCE1 (0.38) MAPTKMT2AMEN1STAT3
SCHEMBL20308912 0.83 RCE1 (0.38) MAPTKMT2AMEN1STAT3
SCHEMBL18241055 0.79 MAPT (0.58) MAPTKMT2AMEN1HIF1ARAB9A
SCHEMBL19672981 0.78 CA1 (0.39) SOS1MAPTKMT2AMEN1STAT3
SCHEMBL19672979 0.78 CA1 (0.39) SOS1MAPTKMT2AMEN1STAT3
SCHEMBL16014387 0.78 MAPT (0.49) MAPTKMT2AMEN1HIF1ASTAT3
SCHEMBL17811450 0.77 MAPT (0.51) MAPTKMT2AMEN1HIF1ARAB9A
SCHEMBL20308925 0.76 TP53 (0.36) SOS1KRASMAPTKMT2AMEN1
SCHEMBL20308929 0.76 CCNE2 (0.33) MAPTKMT2AMEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3252033-B1 TWO-STAGE SYNTHESIS OF N BIARYL COMPOUNDS EVONIK DEGUSSA GMBH (DE) 2018-06-27 EP disclosed