SCHEMBL20327072

SCHEMBL20327072

CN1CCN(C(=O)C2CCC(N)CC2)CC1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.68
LMNA P02545 1/20 0.61
ALDH1A1 P00352 2/20 0.50
TSHR P16473 1/20 0.50
HPGD P15428 1/20 0.50
CHRNB2 P17787 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA4 P43681 1/20 0.47
CHRNB3 Q05901 1/20 0.47
CHRNA6 Q15825 1/20 0.47
HSD11B1 P28845 3/20 0.47
PPP5C P53041 2/20 0.44
PPP2CA P67775 1/20 0.44
TFPI2 P48307 1/20 0.44
NPY4R P50391 1/20 0.44
CYP1A2 P05177 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8252217 1.00 HTT (0.68) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL2688841 0.90 ALDH1A1 (0.60) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL2075903 0.90 HTT (0.81) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL16134884 0.89 HTT (0.59) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL19651225 0.85 HTT (0.53) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL8194135 0.84 HTT (0.71) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL15199119 0.82 HTT (0.70) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL14409695 0.82 HTT (0.70) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL18390863 0.82 HTT (0.70) HTTLMNAALDH1A1TSHRHPGD
SCHEMBL15075709 0.82 HTT (0.55) HTTLMNAALDH1A1TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3558979-B1 NOVEL BENZYLAMINO SUBSTITUTED QUINAZOLINES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-02-17 EP disclosed
WO-2018115380-A1 NOVEL BENZYLAMINO SUBSTITUTED QUINAZOLINES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-06-28 WO disclosed