SCHEMBL20333356

SCHEMBL20333356

O=C1O[C@@H](Cn2nccn2)CN1c1cc(F)c(N2CC[S+]([O-])CC2)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOA P21397 13/20 0.44
CALML3 P27482 3/20 0.43
MAOB P27338 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 1/20 0.40
KCNH2 Q12809 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18410528 0.87 MAOB (0.57) MAOACALML3MAOBKCNH2
SCHEMBL18410621 0.85 MAOA (0.60) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL18410531 0.85 MAOA (0.60) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL18410652 0.85 MAOA (0.48) MAOACALML3MAOBCYP3A4CYP2D6
SCHEMBL18408849 0.85 MAOA (0.48) MAOACALML3MAOBCYP3A4CYP2D6
SCHEMBL18408843 0.85 CALML3 (0.41) MAOACALML3MAOBCYP3A4CYP2D6
SCHEMBL24296584 0.84 CALML3 (0.51) MAOACALML3MAOBCYP3A4
SCHEMBL4015562 0.84 MAOA (0.50) MAOACALML3MAOB
SCHEMBL4017066 0.83 MAOA (0.58) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL18396817 0.83 MAOB (0.54) MAOACALML3MAOBCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3932917-A2 SUBSTITUTED PHENYLOXAZOLIDINONES FOR ANTIMICROBIAL THERAPY The Global Alliance for TB Drug Development, Inc. (US) 2022-01-05 EP disclosed
US-20200148651-A1 SUBSTITUTED PHENYLOXAZOLIDINONES FOR ANTIMICROBIAL THERAPY GLOBAL ALLIANCE FOR TB DRUG DEVELOPMENT INC (US) 2020-05-14 US disclosed
US-10550092-B2 Substituted phenyloxazolidinones for antimicrobial therapy THE GLOBAL ALLIANCE FOR TB DRUG DEVELOPMENT, INC. (US) 2020-02-04 US disclosed
US-20180179168-A1 SUBSTITUTED PHENYLOXAZOLIDINONES FOR ANTIMICROBIAL THERAPY THE GLOBAL ALLIANCE FOR TB DRUG DEVELOPMENT, INC. 2018-06-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180179168-A1 SUBSTITUTED PHENYLOXAZOLIDINONES FOR ANTIMICROBIAL THERAPY THPO, TBCD, OXA1L MAOA 2234/4885CALML3 4026/4885MAOB 1541/4885
US-20200148651-A1 SUBSTITUTED PHENYLOXAZOLIDINONES FOR ANTIMICROBIAL THERAPY THPO, TBCD, OXA1L MAOA 2234/4885CALML3 4026/4885MAOB 1541/4885
US-10550092-B2 Substituted phenyloxazolidinones for antimicrobial therapy THPO, TBCD, OXA1L MAOA 2234/4885CALML3 4026/4885MAOB 1541/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.