SCHEMBL20334459

SCHEMBL20334459

Cc1cc(C)c(CNC=O)c(=O)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EZH2 Q15910 15/20 0.43
EED O75530 7/20 0.43
RBBP4 Q09028 7/20 0.43
SUZ12 Q15022 7/20 0.43
AEBP2 Q6ZN18 7/20 0.43
MAPK1 P28482 1/20 0.40
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20317506 0.81 EZH2 (0.43) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL12684392 0.80 EZH2 (0.49) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL19054922 0.79 EZH2 (0.46) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL20111734 0.79 EZH2 (0.45) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL17885416 0.79 EZH2 (0.48) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL19620987 0.79 KDM4E (0.39) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL19964552 0.77 EZH2 (0.47) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL17788461 0.76 EZH2 (0.46) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL15173371 0.76 EZH2 (0.56) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL19194554 0.75 EZH2 (0.54) EZH2EEDRBBP4SUZ12AEBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323820-B1 SUBSTITUTED 6,5-FUSED BICYCLIC HETEROARYL COMPOUNDS EPIZYME INC (US) 2023-05-10 EP disclosed
WO-2018119357-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ENHANCER OF ZESTE HOMOLOG 2 POLYPEPTIDE Arvinas, Inc. (US) 2018-06-28 WO disclosed