SCHEMBL20338484

SCHEMBL20338484

CS(=O)(=O)C1(Cl)C=Cc2ccccc2N1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
P2RX4 Q99571 1/20 0.32
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904681 0.73 GAA (0.46) GAAMAPT
SCHEMBL6607968 0.73 GAA (0.46) GAAMAPTALDH1A1
SCHEMBL20338456 0.69 MAPT (0.42) GAAMAPTSMN1; SMN2
SCHEMBL2255782 0.69 MAPT (0.50) GAAMAPTP2RX4ALDH1A1SMN1; SMN2
SCHEMBL29789697 0.69 MAPT (0.50) GAAMAPTP2RX4ALDH1A1SMN1; SMN2
SCHEMBL7597347 0.68 GAA (0.37) GAAMAPTP2RX4
SCHEMBL9293762 0.67 GAA (0.43) GAAMAPT
SCHEMBL20338470 0.67 GAA (0.39) GAAMAPT
SCHEMBL21145451 0.66 GAA (0.46) GAAMAPTALDH1A1
SCHEMBL1285713 0.66 MAPT (0.46) GAAMAPTP2RX4ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11464770-B2 Anticancer pharmaceutical composition KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2022-10-11 US disclosed
US-20210315879-A1 ANTICANCER PHARMACEUTICAL COMPOSITION NATIONAL CANCER CENTER (KR) 2021-10-14 US disclosed
US-10227306-B2 Compounds for inhibiting c-myc/max/DNA complex formation NATIONAL CANCER CENTER (KR) 2019-03-12 US disclosed
US-20180186744-A1 COMPOUNDS FOR INHIBITING C-MYC/MAX/DNA COMPLEX FORMATION NATIONAL CANCER CENTER (KR) 2018-07-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11464770-B2 Anticancer pharmaceutical composition MYC, MYCBP, TP53 GAA 1125/4885MAPT 848/4885P2RX4 4873/4885
US-10227306-B2 Compounds for inhibiting c-myc/max/DNA complex formation MYC, MYCBP, MYCBP2 GAA 1908/4885MAPT 2894/4885P2RX4 4876/4885
US-20180186744-A1 COMPOUNDS FOR INHIBITING C-MYC/MAX/DNA COMPLEX FORMATION MYC, MYCBP, MYCBP2 GAA 1908/4885MAPT 2894/4885P2RX4 4876/4885
US-20210315879-A1 ANTICANCER PHARMACEUTICAL COMPOSITION MYC, MYCBP, TP53 GAA 1125/4885MAPT 848/4885P2RX4 4873/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.