SCHEMBL20339529

SCHEMBL20339529

Cc1ccnc(N2CCN(C(=O)O)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.51
HPGD P15428 1/20 0.51
PARP1 P09874 1/20 0.51
CPT2 P23786 1/20 0.50
CPT1A P50416 1/20 0.50
CPT1B Q92523 1/20 0.50
ALDH1A1 P00352 5/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HSD17B10 Q99714 2/20 0.48
HTT P42858 2/20 0.48
TSHR P16473 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAPT P10636 1/20 0.48
GRIN2D O15399 1/20 0.48
GRIN3B O60391 1/20 0.48
GRIN1 Q05586 1/20 0.48
GRIN2A Q12879 1/20 0.48
GRIN2B Q13224 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15286922 0.94 PROKR1 (0.51) KDM4EHPGDPARP1CPT2CPT1A
SCHEMBL15450884 0.88 KDM4E (0.51) KDM4EHPGDPARP1CPT2CPT1A
SCHEMBL18949715 0.85 GRIN2D (0.60) KDM4EHPGDALDH1A1HSD17B10HTT
SCHEMBL15228566 0.84 PIK3CA (0.48) KDM4EHPGDALDH1A1SMN1; SMN2HSD17B10
SCHEMBL19998582 0.82 USP30 (0.52) KDM4EHPGDCPT2CPT1ACPT1B
SCHEMBL30525303 0.81 OPRD1 (0.55) KDM4EHPGDALDH1A1HSD17B10GRIN2D
SCHEMBL28772301 0.81 GRM5 (0.60) KDM4EHPGDALDH1A1SMN1; SMN2HSD17B10
SCHEMBL322198 0.81 KMT2A (0.48) KDM4EHPGDALDH1A1SMN1; SMN2HSD17B10
SCHEMBL390627 0.81 HRH3 (0.57) KDM4EHPGDALDH1A1HSD17B10HTT
SCHEMBL16795243 0.81 GRIN2D (0.51) KDM4EHPGDALDH1A1SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3562822-A1 POLY-ADP RIBOSE POLYMERASE (PARP) INHIBITORS Mitobridge, Inc. (US) 2019-11-06 EP disclosed
WO-2018125961-A1 POLY-ADP RIBOSE POLYMERASE (PARP) INHIBITORS MITOBRIDGE, INC. (US) 2018-07-05 WO disclosed
CN-102803225-A Imidazole derivatives and their use as modulators of cyclin dependent kinases NOVARTIS AG 2012-11-28 CN disclosed