SCHEMBL20342425

SCHEMBL20342425

COCc1cncc(-n2cnnn2)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.44
MAPT P10636 3/20 0.40
TP53 P04637 1/20 0.40
HTT P42858 2/20 0.38
GAA P10253 2/20 0.38
KCNH2 Q12809 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 5/20 0.37
LMNA P02545 1/20 0.37
ABL1 P00519 1/20 0.37
RIN1 Q13671 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
F2 P00734 1/20 0.37
KCNJ1 P48048 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19381177 0.80 NOTUM (0.45) NOTUMMAPTTP53HTTKCNH2
SCHEMBL20342502 0.79 TP53 (0.56) NOTUMTP53LMNATSHRKMT2A
SCHEMBL18216595 0.78 MAPT (0.58) NOTUMMAPTHTTGAAKDM4E
SCHEMBL16122139 0.77 NOTUM (0.41) NOTUMMAPTTP53HTTGAA
SCHEMBL15018021 0.75 KMT2A (0.45) NOTUMMAPTTP53GAAKCNH2
SCHEMBL17858623 0.74 NOTUM (0.67) NOTUMMAPTHTTALDH1A1LMNA
SCHEMBL18216598 0.74 NOTUM (0.45) NOTUMMAPTTP53HTTGAA
SCHEMBL18216589 0.73 GPR119 (0.43) NOTUMMAPTHTTGAAKDM4E
SCHEMBL19381035 0.73 MAPT (0.47) NOTUMMAPTTP53HTTGAA
SCHEMBL19381199 0.72 GPR119 (0.43) NOTUMALDH1A1F2KCNJ1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968288-B1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME (US) 2018-07-04 EP disclosed