SCHEMBL20344302

SCHEMBL20344302

c1ccc(C(C[C@H]2CCCN2)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.51
CACNA2D1 P54289 1/20 0.49
CACNA1B Q00975 1/20 0.49
CACNB1 Q02641 1/20 0.49
LTA4H P09960 4/20 0.45
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CYP2D6 P10635 1/20 0.44
HTR6 P50406 2/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8493732 0.95 POLB (0.59) POLBCACNA2D1CACNA1BCACNB1LTA4H
SCHEMBL22259900 0.84 CYP2D6 (0.56) POLBCACNA2D1CACNA1BCACNB1CYP2D6
SCHEMBL8507267 0.84 CYP2D6 (0.56) POLBCACNA2D1CACNA1BCACNB1CYP2D6
SCHEMBL20833013 0.84 CYP2D6 (0.56) POLBCACNA2D1CACNA1BCACNB1CYP2D6
SCHEMBL3582733 0.84 POLB (0.47) POLBCACNA2D1CACNA1BCACNB1LTA4H
SCHEMBL11447515 0.84 POLB (0.47) POLBCACNA2D1CACNA1BCACNB1LTA4H
SCHEMBL20832991 0.84 CYP2D6 (0.56) POLBCACNA2D1CACNA1BCACNB1CYP2D6
SCHEMBL6535642 0.82 CHRNB4 (0.49) POLBLTA4HCHRNB4CHRNA3SLC6A2
SCHEMBL10681797 0.80 POLB (0.54) POLBCACNA2D1CACNA1BCACNB1LTA4H
SCHEMBL10679403 0.80 CYP2D6 (0.62) POLBCACNA2D1CACNA1BCACNB1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2792664-B1 OPTICAL RESOLUTION METHOD FOR BICYCLIC COMPOUND USING ASYMMETRIC CATALYST DAIICHI SANKYO CO LTD (JP) 2018-07-04 EP disclosed