SCHEMBL20344687

SCHEMBL20344687

COc1cc(OCC(C)C)ccc1-c1ccc2c(c1COc1cc(F)ccc1C)N(C)C(=O)C(C)(C)N2

nearest known ligand 0.88

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IL6 P05231 8/20 0.88
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
PLA2G7 Q13093 1/20 0.32
HTR2C P28335 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
MDM2 Q00987 1/20 0.31
CTSD P07339 1/20 0.31
BACE1 P56817 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20335196 0.94 IL6 (1.00) IL6PLA2G7HTR2CMDM2ALDH1A1
SCHEMBL18573526 0.94 IL6 (1.00) IL6PLA2G7HTR2CMDM2ALDH1A1
SCHEMBL18573562 0.94 IL6 (1.00) IL6PLA2G7HTR2CMDM2ALDH1A1
SCHEMBL4581163 0.92 IL6 (0.82) IL6PLA2G7HTR2CMDM2ALDH1A1
SCHEMBL20344710 0.92 IL6 (0.82) IL6PLA2G7
SCHEMBL18573466 0.92 IL6 (0.90) IL6ALDH1A1MAPK1
SCHEMBL20335223 0.92 IL6 (1.00) IL6ALDH1A1MAPK1
SCHEMBL18573599 0.92 IL6 (1.00) IL6ALDH1A1MAPK1
SCHEMBL18573549 0.92 IL6 (1.00) IL6ALDH1A1MAPK1
SCHEMBL20344621 0.91 IL6 (0.83) IL6PLA2G7HTR2CMDM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3342768-A1 [4-(1, 3, 3-TRIMETHYL-2-OXO-3, 4-DIHYDRO-1H-QUINOXALIN-7-YL) PHENOXY]ETHYLOXY COMPOUND OR SALT THEREOF Santen Pharmaceutical Co., Ltd. (JP) 2018-07-04 EP disclosed