SCHEMBL20345733

SCHEMBL20345733

COCc1nnc(N2CC3CC3C2)n1-c1ccc(OC)nc1

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OXTR P30559 10/20 0.68
AVPR1A P37288 15/20 0.66
AVPR2 P30518 11/20 0.63
AVPR1B P47901 7/20 0.62
TACR1 P25103 1/20 0.62
OPRK1 P41145 1/20 0.62
GHSR Q92847 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4124946 0.89 AVPR1A (0.66) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL4112837 0.83 AVPR1A (0.65) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL8271860 0.83 AVPR1A (0.67) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL4125784 0.83 AVPR1A (0.67) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL4111772 0.82 AVPR1A (0.68) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL4132742 0.79 AVPR1A (0.76) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL4118198 0.79 OXTR (0.72) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL4118667 0.78 OXTR (0.68) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL20327957 0.78 AVPR1A (1.00) OXTRAVPR1AAVPR2AVPR1BTACR1
SCHEMBL20327922 0.77 AVPR1A (0.75) OXTRAVPR1AAVPR2AVPR1BTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3564231-A1 AZABICYCLO-SUBSTITUTED TRIAZOLE DERIVATIVE, PREPARATION METHOD THEREOF, AND APPLICATION OF SAME IN MEDICINE Jiangsu Hengrui Medicine Co., Ltd. (CN) 2019-11-06 EP disclosed
WO-2018121551-A1 AZABICYCLO-SUBSTITUTED TRIAZOLE DERIVATIVE, PREPARATION METHOD THEREOF, AND APPLICATION OF SAME IN MEDICINE 江苏恒瑞医药股份有限公司 2018-07-05 WO disclosed