SCHEMBL20376337

SCHEMBL20376337

CS(=O)(=O)c1nc(C(N)=O)c(-c2ccc(F)cc2)[nH]1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.58
PTGS1 P23219 6/20 0.58
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
CDC7 O00311 1/20 0.44
MAPK14 Q16539 2/20 0.41
ALOX5 P09917 1/20 0.41
CSNK1A1 P48729 1/20 0.41
CSNK1D P48730 1/20 0.41
CSNK1E P49674 1/20 0.41
MAPK11 Q15759 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CSNK1A1L Q8N752 1/20 0.41
GSK3B P49841 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30879827 0.91 PTGS2 (0.54) PTGS2PTGS1ALDH1A1HPGDCDC7
SCHEMBL18161744 0.89 PTGS2 (0.58) PTGS2PTGS1ALDH1A1HPGDMAPK14
SCHEMBL14692607 0.87 PTGS2 (0.59) PTGS2PTGS1ALDH1A1HPGDMAPK14
SCHEMBL14692454 0.84 PTGS2 (0.59) PTGS2PTGS1ALDH1A1HPGDMAPK14
SCHEMBL22068721 0.72 PTGS1 (0.78) PTGS2PTGS1ALDH1A1HPGDMAPK14
SCHEMBL3120716 0.72 MAPK13 (0.57) PTGS2ALDH1A1HPGDCDC7MAPK14
SCHEMBL4467134 0.71 MAPK14 (0.63) PTGS2PTGS1MAPK14GSK3B
SCHEMBL14692202 0.70 PTGS2 (0.63) PTGS2PTGS1ALDH1A1HPGDMAPK14
SCHEMBL30879817 0.69 MAPK14 (0.51) PTGS2PTGS1MAPK14MAPK11GSK3B
SCHEMBL30879822 0.66 CDC7 (0.38) PTGS2PTGS1ALDH1A1CDC7MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2739143-B1 PREPARATION AND METHODS OF USE FOR ORTHO-ARYL 5- MEMBERED HETEROARYL-CARBOXAMIDE CONTAINING MULTI-TARGETED KINASE INHIBITORS FLYNN GARY A (US) 2018-07-11 EP disclosed