SCHEMBL20389256

SCHEMBL20389256

Cc1ccc2c(c1)CCN(S(=O)(=O)c1ccc(N)cc1)C2

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.60
ESR2 Q92731 2/20 0.53
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
PKM P14618 3/20 0.51
CD4 P01730 3/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
LMNA P02545 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
ESR1 P03372 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14751054 0.92 AKR1C3 (0.65) AKR1C3ESR2MEN1KMT2APKM
SCHEMBL1949180 0.83 PKM (0.54) MEN1KMT2APKMSMN1; SMN2LMNA
SCHEMBL15122772 0.83 AKR1C3 (0.74) AKR1C3SMN1; SMN2LMNA
SCHEMBL20389408 0.81 KMT2A (0.77) AKR1C3ESR2MEN1KMT2ACYP3A4
SCHEMBL5632531 0.81 AKR1C3 (0.60) AKR1C3ESR2MEN1KMT2APKM
SCHEMBL2590065 0.81 AKR1C3 (0.60) AKR1C3ESR2MEN1KMT2APKM
SCHEMBL20910236 0.81 CA7 (0.58) AKR1C3ESR2MEN1KMT2APKM
SCHEMBL15122441 0.79 AKR1C3 (0.73) AKR1C3SMN1; SMN2LMNA
SCHEMBL13302259 0.79 KMT2A (0.77) AKR1C3MEN1KMT2APKMCYP3A4
SCHEMBL13102503 0.78 ESR2 (0.69) AKR1C3ESR2MEN1KMT2ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018132372-A1 SMALL MOLECULE ACTIVATORS OF NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE (NAMPT) AND USES THEREOF Sanford Burnham Prebys Medical Discovery Institute (US) 2018-07-19 WO disclosed