SCHEMBL20394258

SCHEMBL20394258

Cc1nsc(C)c1-c1cccnc1Oc1ccc(C(C)(F)F)nc1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 5/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
ATM Q13315 1/20 0.33
PDE10A Q9Y233 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20394339 0.80 BRD4 (0.40) DRD1ALDH1A1
SCHEMBL18661513 0.79 PDE10A (0.42) PDE10A
SCHEMBL20394248 0.78 BRD4 (0.37) DRD1ALDH1A1PDE10A
SCHEMBL20406568 0.77 DRD1 (0.38) DRD1ALDH1A1MAPTATM
SCHEMBL20394327 0.76 CYP17A1 (0.38) DRD1PDE10A
SCHEMBL20406275 0.76 PDE10A (0.38) DRD1PDE10A
SCHEMBL18661454 0.76 PDE10A (0.35) DRD1PDE10A
SCHEMBL20394511 0.75 PDE10A (0.34) DRD1ALDH1A1MAPTATMPDE10A
SCHEMBL18661516 0.75 PDE10A (0.45) ALDH1A1PDE10A
SCHEMBL20406785 0.75 DRD1 (0.38) DRD1MAPTPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3351533-B1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME KAKEN PHARMA CO LTD (JP) 2025-07-23 EP disclosed
US-10647675-B2 Biaryl derivative and medicine containing same KAKEN PHARMACEUTICAL CO., LTD. (JP) 2020-05-12 US disclosed
US-20190055199-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME KAKEN PHARMACEUTICAL CO., LTD. (JP) 2019-02-21 US disclosed
EP-3351533-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME Kaken Pharmaceutical Co., Ltd. (JP) 2018-07-25 EP disclosed
EP-3351533-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME Kaken Pharmaceutical Co., Ltd. (JP) 2018-07-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10647675-B2 Biaryl derivative and medicine containing same MAN2B1, CBR3, MANBA DRD1 1032/4885ALDH1A1 2994/4885MAPT 4703/4885
US-20190055199-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME MAN2B1, CBR3, MANBA DRD1 1032/4885ALDH1A1 2994/4885MAPT 4703/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.