SCHEMBL20394265

SCHEMBL20394265

COc1c(Cl)cncc1-c1cccnc1Oc1ccc(C(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 3/20 0.42
LMNA P02545 1/20 0.40
AHR P35869 1/20 0.40
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
GPBAR1 Q8TDU6 1/20 0.39
MCHR1 Q99705 1/20 0.39
PDE10A Q9Y233 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20394356 0.93 PDE10A (0.38) NPBWR1KMT2APDE10A
SCHEMBL18661523 0.88 AHR (0.40) AHRGPBAR1PDE10A
SCHEMBL20394428 0.87 NPBWR1 (0.42) NPBWR1LMNAKMT2AATMMCHR1
SCHEMBL18661345 0.85 PDE10A (0.38) PDE10A
SCHEMBL18661519 0.84 ABL1 (0.36) LMNAGPBAR1PDE10A
SCHEMBL20394232 0.84 MAPT (0.44) NPBWR1MCHR1PDE10A
SCHEMBL20394208 0.82 PDE10A (0.49) AHRGPBAR1PDE10A
SCHEMBL20406748 0.82 PDE10A (0.38) KMT2APDE10A
SCHEMBL20394494 0.82 PDE10A (0.38) KMT2APDE10A
SCHEMBL20394256 0.81 FEN1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3351533-B1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME KAKEN PHARMA CO LTD (JP) 2025-07-23 EP disclosed
US-10647675-B2 Biaryl derivative and medicine containing same KAKEN PHARMACEUTICAL CO., LTD. (JP) 2020-05-12 US disclosed
US-10647675-B2 Biaryl derivative and medicine containing same KAKEN PHARMACEUTICAL CO., LTD. (JP) 2020-05-12 US disclosed
US-20190055199-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME KAKEN PHARMACEUTICAL CO., LTD. (JP) 2019-02-21 US disclosed
US-20190055199-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME KAKEN PHARMACEUTICAL CO., LTD. (JP) 2019-02-21 US disclosed
EP-3351533-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME Kaken Pharmaceutical Co., Ltd. (JP) 2018-07-25 EP disclosed
EP-3351533-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME Kaken Pharmaceutical Co., Ltd. (JP) 2018-07-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10647675-B2 Biaryl derivative and medicine containing same MAN2B1, CBR3, MANBA NPBWR1 1051/4885LMNA 1952/4885AHR 38/4885
US-20190055199-A1 BIARYL DERIVATIVE AND MEDICINE CONTAINING SAME MAN2B1, CBR3, MANBA NPBWR1 1051/4885LMNA 1952/4885AHR 38/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.