SCHEMBL20401464

SCHEMBL20401464

COc1ccc(Cn2ncc3cc(N)ccc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 1/20 0.48
QPCTL Q9NXS2 1/20 0.48
NPBWR1 P48145 6/20 0.47
BRD4 O60885 1/20 0.46
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
EGFR P00533 3/20 0.44
ERBB2 P04626 3/20 0.44
CACNA1H O95180 1/20 0.43
MCHR1 Q99705 1/20 0.43
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
RECQL P46063 1/20 0.43
DCTPP1 Q9H773 1/20 0.43
PDE1A P54750 1/20 0.43
PDE1B Q01064 1/20 0.43
PDE1C Q14123 1/20 0.43
CHEK1 O14757 1/20 0.43
AURKA O14965 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29447767 1.00 QPCT (0.48) QPCTQPCTLNPBWR1BRD4HTR2A
SCHEMBL24996626 0.86 QPCT (0.46) QPCTQPCTLNPBWR1BRD4EGFR
SCHEMBL30879444 0.86 QPCT (0.46) QPCTQPCTLNPBWR1BRD4EGFR
SCHEMBL3379521 0.86 EGFR (0.57) QPCTQPCTLEGFRERBB2RECQL
SCHEMBL3538945 0.84 RECQL (0.51) EGFRERBB2MCHR1GRIN1GRIN2B
SCHEMBL10080163 0.84 NPBWR1 (0.47) QPCTQPCTLNPBWR1BRD4HTR2A
SCHEMBL2443709 0.84 NPBWR1 (0.47) QPCTQPCTLNPBWR1BRD4HTR2A
SCHEMBL24996628 0.84 NPBWR1 (0.47) QPCTQPCTLNPBWR1BRD4HTR2A
SCHEMBL30879430 0.84 NPBWR1 (0.47) QPCTQPCTLNPBWR1BRD4HTR2A
SCHEMBL530059 0.84 IDO1 (0.47) QPCTQPCTLNPBWR1BRD4ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018136935-A1 2-ARYLSULFONAMIDO-N-ARYLACETAMIDE DERIVATIZED STAT3 INHIBITORS UNIVERSITY OF HAWAII (US) 2018-07-26 WO disclosed
WO-2018136935-A1 2-ARYLSULFONAMIDO-N-ARYLACETAMIDE DERIVATIZED STAT3 INHIBITORS UNIVERSITY OF HAWAII (US) 2018-07-26 WO disclosed