SCHEMBL20404396

SCHEMBL20404396

CCc1nc2cccc(C)c2c(=O)n1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 5/20 0.57
PIK3R1 P27986 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.52
ALDH1A1 P00352 1/20 0.52
PIK3CG P48736 1/20 0.50
ESR1 P03372 1/20 0.49
ESR2 Q92731 1/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.46
MAPT P10636 1/20 0.46
USP2 O75604 1/20 0.45
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
KCNH2 Q12809 2/20 0.45
HRH3 Q9Y5N1 2/20 0.45
PSMD14 O00487 1/20 0.44
POLB P06746 1/20 0.44
RECQL P46063 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21028899 0.91 PIK3CD (0.60) PIK3CDPIK3R1SMN1; SMN2ALDH1A1PIK3CG
SCHEMBL358165 0.89 PIK3CD (0.62) PIK3CDPIK3R1SMN1; SMN2ALDH1A1PIK3CG
SCHEMBL20081323 0.88 PIK3CD (0.51) PIK3CDPIK3R1SMN1; SMN2ALDH1A1PIK3CG
SCHEMBL15817691 0.87 PIK3CD (0.77) PIK3CDPIK3R1SMN1; SMN2ALDH1A1PIK3CG
SCHEMBL16597182 0.86 SMN1; SMN2 (0.50) PIK3CDPIK3R1SMN1; SMN2ALDH1A1PIK3CG
SCHEMBL17235505 0.86 ESR1 (0.60) SMN1; SMN2ALDH1A1ESR1ESR2NPC1
SCHEMBL16597185 0.86 PDE10A (0.52) PIK3CDPIK3R1SMN1; SMN2ALDH1A1PIK3CG
SCHEMBL9604076 0.86 PIK3CD (0.76) PIK3CDPIK3R1ALDH1A1PIK3CGL3MBTL1
SCHEMBL22237904 0.85 PIK3CD (0.50) PIK3CDPIK3R1SMN1; SMN2ALDH1A1PIK3CG
SCHEMBL15864426 0.84 PIK3CD (0.67) PIK3CDPIK3R1PIK3CGNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935246-B1 ISOQUINOLINONE OR QUINAZOLINONE PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD CALISTOGA LLC (US) 2018-07-25 EP disclosed