SCHEMBL20406038

SCHEMBL20406038

OC[C@@H]1CN(Cc2ccc(-c3noc(-c4nnn(-c5ccccc5F)c4-c4ccncc4)n3)cc2)CCO1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.40
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
S1PR4 O95977 1/20 0.38
S1PR5 Q9H228 1/20 0.38
S1PR3 Q99500 7/20 0.37
KCNH2 Q12809 1/20 0.37
NPC1 O15118 1/20 0.36
PKM P14618 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
DRD4 P21917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3760963 1.00 S1PR1 (0.40) S1PR1HDAC8HDAC6S1PR4S1PR5
SCHEMBL3751149 0.88 ALOX5 (0.43) S1PR1HDAC6KCNH2NPC1PKM
SCHEMBL3751157 0.87 CYP2D6 (0.45) S1PR1
SCHEMBL3761101 0.87 S1PR1 (0.41) S1PR1S1PR4S1PR5S1PR3KCNH2
SCHEMBL3750299 0.87 S1PR1 (0.41) S1PR1S1PR4S1PR5S1PR3NPC1
SCHEMBL3755464 0.87 S1PR1 (0.41) S1PR1S1PR4S1PR5S1PR3KCNH2
SCHEMBL3748523 0.87 S1PR1 (0.41) S1PR1S1PR4S1PR5S1PR3KCNH2
SCHEMBL13765565 0.87 S1PR1 (0.41) S1PR1S1PR4S1PR5S1PR3KCNH2
SCHEMBL3762551 0.87 S1PR1 (0.43) S1PR1S1PR4S1PR5S1PR3KCNH2
SCHEMBL3756948 0.86 S1PR1 (0.45) S1PR1KCNH2NPC1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250165-B1 TRIAZOLE OXADIAZOLES DERIVATIVES MERCK SERONO SA (CH) 2018-07-25 EP disclosed